partial agonist造句

• It is a partial agonist for the benzodiazepine site of the efficacy.
• Pridopidine, therefore, differs from D 2 receptor antagonists, agonists and partial agonists.
• Compounds considered partial agonists tend to have efficacy in between this range.
• Some opioid agonist-antagonists, partial agonists, and inverse agonists are also derived from morphine.
• On the other hand, aripiprazole is a partial agonist of the dopamine receptor.
• "' Bufuralol "'is a potent beta-adrenoceptor antagonist with partial agonist activity.
• It is a partial agonist at the cannabinoid Ki of 8.45nM.
• DOC acts as a selective 5-HT 2C receptor partial agonist.
• RWJ-51204 is a nonselective partial agonist at GABA A receptors.
• Like varenicline, cytisine is a partial agonist of nicotinic acetylcholine receptors ( nAChRs ).
• Pipequaline acts as a non-selective GABA A receptor partial agonist.
• Andarine is an orally active partial agonist for androgen receptors.
• Some ginsenosides have also been shown to be partial agonists of steroid hormone receptors.
• It is a 3rd generation adrenergic ? receptor partial agonist.
• There are inconsistent findings about an additional activity as a dopamine D2 receptor partial agonist.
• Examples of ligands activating peroxisome proliferator-activated receptor gamma as partial agonists are honokiol and falcarindiol.
• Cariprazine has partial agonist as well as antagonist properties depending on the endogenous dopamine levels.
• "' Ipsapirone "'is a 5-HT 1A receptor partial agonist of the piperazine and azapirone chemical classes.
• Sameridine has an unusual pharmacological profile, being both a local anaesthetic and a ?-opioid partial agonist.
• It acts as a partial agonist of the opioid receptors, with mixed agonist and antagonist effects.